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(350) Indirect Publications in 2009

Abdul-Ghani, R., Loutfy, N., Sahn, A. E., & Hassan, A. (2009). Current chemotherapy arsenal for schistosomiasis mansoni: Alternatives and challenges. Parasitology Research, 104(5), 955-965.

Abdul-Ghani, R. A., Loutfy, N., & Hassan, A. (2009). Experimentally promising antischistosomal drugs: A review of some drug candidates not reaching the clinical use. Parasitology Research, 105(4), 899-906.

Abulafia, D. P., De Rivero Vaccari, J. P., Lozano, J. D., Lotocki, G., Keane, R. W., & Dietrich, W. D. (2009). Inhibition of the inflammasome complex reduces the inflammatory response after thromboembolic stroke in mice. Journal of Cerebral Blood Flow and Metabolism, 29(3), 534-544.

Allgeier, S. H., Vezina, C. M., Lin, T. -., Moore, R. W., Silverstone, A. E., Mukai, M., et al. (2009). Estrogen signaling is not required for prostatic bud patterning or for its disruption by 2,3,7,8-tetrachlorodibenzo-p-dioxin. Toxicology and Applied Pharmacology, 239(1), 80-86.

Ananthan, S., Zhang, W., & Hobrath, J. V. (2009). Recent advances in structure-based virtual screening of G-protein coupled receptors. AAPS Journal, 11(1), 178-185.

Andersen, M. E., & Krewski, D. (2009). Toxicity testing in the 21st century: Bringing the vision to life. Toxicological Sciences, 107(2), 324-330.

Angelopoulos, N., Hadjiprocopis, A., & Walkinshaw, M. D. (2009). Bayesian model averaging for ligand discovery. Journal of Chemical Information and Modeling, 49(6), 1547-1557.

Antony, J., Kellershohn, K., Mohr-Andrä, M., Kebig, A., Prilla, S., Muth, M., et al. (2009). Dualsteric GPCR targeting: A novel route to binding and signaling pathway selectivity. FASEB Journal, 23(2), 442-450.

Arkin, M. R., & Whitty, A. (2009). The road less traveled: Modulating signal transduction enzymes by inhibiting their protein-protein interactions. Current Opinion in Chemical Biology, 13(3), 284-290.

Auld, D. S., Zhang, Y. -., Southall, N. T., Rai, G., Landsman, M., MacLure, J., et al. (2009). A basis for reduced chemical library inhibition of firefly luciferase obtained from directed evolution. Journal of Medicinal Chemistry, 52(5), 1450-1458.

Bachovchin, D. A., Brown, S. J., Rosen, H., & Cravatt, B. F. (2009). Identification of selective inhibitors of uncharacterized enzymes by high-throughput screening with fluorescent activity-based probes. Nature Biotechnology, 27(4), 387-394.

Barton, M., & Meyer, M. R. (2009). Postmenopausal hypertension: Mechanisms and therapy. Hypertension, 54(1), 11-18.

Baškovč, J., Bevk, D., Stanovnik, B., & Svete, J. (2009). Bis-enaminone based parallel solution-phase synthesis of 1,4-dihydropyridine derivatives. Journal of Combinatorial Chemistry, 11(3), 500-507.

Baxendale, I. R., Ley, S. V., Mansfield, A. C., & Smith, C. D. (2009). Multistep synthesis using modular flow reactors: Bestmann-ohira reagent for the formation of alkynes and triazoles. Angewandte Chemie – International Edition, 48(22), 4017-4021.

Bayne, C. J. (2009). Successful parasitism of vector snail biomphalaria glabrata by the human blood fluke (trematode) schistosoma mansoni: A 2009 assessment. Molecular and Biochemical Parasitology, 165(1), 8-18.

Bergsbaken, T., Fink, S. L., & Cookson, B. T. (2009). Pyroptosis: Host cell death and inflammation. Nature Reviews Microbiology, 7(2), 99-109.

Berrodin, T. J., Chang, K. C. N., Komm, B. S., Freedman, L. P., & Nagpal, S. (2009). Differential biochemical and cellular actions of premarin estrogens: Distinct pharmacology of bazedoxifene-conjugated estrogens combination. Molecular Endocrinology, 23(1), 74-85.

Bharate, S. B., Nemmani, K. V. S., & Vishwakarma, R. A. (2009). Progress in the discovery and development of small-molecule modulators of G-protein-coupled receptor 40 (GPR40/FFA1/FFAR1): An emerging target for type 2 diabetes. Expert Opinion on Therapeutic Patents, 19(2), 237-264.

Bickel, P. E., Tansey, J. T., & Welte, M. A. (2009). PAT proteins, an ancient family of lipid droplet proteins that regulate cellular lipid stores. Biochimica Et Biophysica Acta – Molecular and Cell Biology of Lipids, 1791(6), 419-440.

Biersack, B., & Schobert, R. (2009). Metallodrug conjugates with steroids and selective estrogen receptor modulators (SERM). Current Medicinal Chemistry, 16(18), 2324-2337.

Biffinger, J., Ribbens, M., Ringeisen, B., Pietron, J., Finkel, S., & Nealson, K. (2009). Characterization of electrochemically active bacteria utilizing a high-throughput voltage-based screening assay. Biotechnology and Bioengineering, 102(2), 436-444.

Blackburn, W. H., Dickerson, E. B., Smith, M. H., McDonald, J. F., & Lyon, L. A. (2009). Peptide-functionalized nanogels for targeted siRNA delivery. Bioconjugate Chemistry, 20(5), 960-968.

Blaskovich, M. A. T. (2009). Drug discovery and protein tyrosine phosphatases. Current Medicinal Chemistry, 16(17), 2095-2176.

Blom, W. M., van Nielen, W. G. L., de Groene, E. M., & Albers, R. (2009). A cell-based screening assay for natural killer cell activity. International Immunopharmacology, 9(6), 746-752.

Blum, L. C., & Reymond, J. -. (2009). 970 million druglike small molecules for virtual screening in the chemical universe database GDB-13. Journal of the American Chemical Society, 131(25), 8732-8733.

Bogdan, A. R., & Sach, N. W. (2009). The use of copper flow reactor technology for the continuous synthesis of 1,4-disubstituted 1,2,3-triazoles. Advanced Synthesis and Catalysis, 351(6), 849-854.

Boisselier, E., & Astruc, D. (2009). Gold nanoparticles in nanomedicine: Preparations, imaging, diagnostics, therapies and toxicity. Chemical Society Reviews, 38(6), 1759-1782.

Bourque, M., Dluzen, D. E., & Di Paolo, T. (2009). Neuroprotective actions of sex steroids in parkinson’s disease. Frontiers in Neuroendocrinology, 30(2), 142-157.

Bouskine, A., Nebout, M., Brücker-Davis, F., Banahmed, M., & Fenichel, P. (2009). Low doses of bisphenol A promote human seminoma cell proliferation by activating PKA and PKG via a membrane G-protein-coupled estrogen receptor. Environmental Health Perspectives, 117(7), 1053-1058.

Brady, L. S., Winsky, L., Goodman, W., Oliveri, M. E., & Stover, E. (2009). NIMH initiatives to facilitate collaborations among industry, academia, and government for the discovery and clinical testing of novel models and drugs for psychiatric disorders. Neuropsychopharmacology, 34(1), 229-243.

Brannan, J. M., Dong, W., Prudkin, L., Behrens, C., Lotan, R., Bekele, B. N., et al. (2009). Expression of the receptor tyrosine kinase EphA2 is increased in smokers and predicts poor survival in non -small cell lung cancer. Clinical Cancer Research, 15(13), 4423-4430.

Brinton, R. D. (2009). Estrogen-induced plasticity from cells to circuits: Predictions for cognitive function. Trends in Pharmacological Sciences, 30(4), 212-222.

Brufani, M., Ceccacci, F., Filocamo, L., Garofalo, B., Joudioux, R., Bella, A. L., et al. (2009). Novel locally active estrogens accelerate cutaneous wound healing. A preliminary study. Molecular Pharmaceutics, 6(2), 543-556.

Bryant, C., & Fitzgerald, K. A. (2009). Molecular mechanisms involved in inflammasome activation. Trends in Cell Biology, 19(9), 455-464.

Burr, I., Winchester, T., Keighley, W., & Sewing, A. (2009). Compound management beyond efficiency. Journal of Biomolecular Screening, 14(5), 485-491.

Caffrey, C. R., Rohwer, A., Oellien, F., Marhöfer, R. J., Braschi, S., Oliveira, G., et al. (2009). A comparative chemogenomics strategy to predict potential drug targets in the metazoan pathogen, schistosoma mansoni. PLoS ONE, 4(2)

Camerer, E., Regard, J. B., Cornelissen, I., Srinivasan, Y., Duong, D. N., Palmer, D., et al. (2009). Sphingosine-1-phosphate in the plasma compartment regulates basal and inflammation-induced vascular leak in mice. Journal of Clinical Investigation, 119(7), 1871-1879.

Campbell, W. C., Conder, G. A., & Marchiondo, A. A. (2009). Future of the animal health industry at a time of food crisis. Veterinary Parasitology, 163(3), 188-195.

Card, A., Caldwell, C., Min, H., Lokchander, B., Xi, H., Sciabola, S., et al. (2009). High-throughput biochemical kinase selectivity assays: Panel development and screening applications. Journal of Biomolecular Screening, 14(1), 31-42.

Castellino, F. J., & Ploplis, V. A. (2009). The protein C pathway and pathologic processes. Journal of Thrombosis and Haemostasis, 7(SUPPL. 1), 140-145.

Chae, J. J., Aksentijevich, I., & Kastner, D. L. (2009). Advances in the understanding of familial mediterranean fever and possibilities for targeted therapy. British Journal of Haematology, 146(5), 467-478.

Chang, E., Congdon, E. E., Honson, N. S., Duff, K. E., & Kuret, J. (2009). Structure-activity relationship of cyanine tau aggregation inhibitors. Journal of Medicinal Chemistry, 52(11), 3539-3547.

Chen, C. -., & Reamer, R. A. (2009). A facile synthesis of N,3-disubstituted indoles and 3-hydroxyl indolines via an intramolecular SNAr of fluorinated amino alcohols. Tetrahedron Letters, 50(14), 1529-1532.

Chen, G., Shaw, M. H., Kim, Y. -., & Nuñez, G. (2009). NOD-like receptors: Role in innate immunity and inflammatory disease

Chu, Z., Andrade, J., Shupnik, M. A., & Moenter, S. M. (2009). Differential regulation of gonadotropin-releasing hormone neuron activity and membrane properties by acutely applied estradiol: Dependence on dose and estrogen receptor subtype. Journal of Neuroscience, 29(17), 5616-5627.

Clapham, K. M., Batsanov, A. S., Bryce, M. R., & Tarbit, B. (2009). Trifluoromethyl-substituted pyridyl- and pyrazolylboronic acids and esters: Synthesis and suzuki-miyaura cross-coupling reactions. Organic and Biomolecular Chemistry, 7(10), 2155-2161.

Clarke, D. L., Dakshinamurti, S., Larsson, A. -., Ward, J. E., & Yamasaki, A. (2009). Lipid metabolites as regulators of airway smooth muscle function. Pulmonary Pharmacology and Therapeutics, 22(5), 426-435.

Codocedo, J. F., Rodríguez, F. E., & Huidobro-Toro, J. P. (2009). Neurosteroids differentially modulate P2X4 ATP-gated channels through non-genomic interactions. Journal of Neurochemistry, 110(2), 734-744.

Coma, I., Clark, L., Diez, E., Harper, G., Herranz, J., Hofmann, G., et al. (2009). Process validation and screen reproducibility in high-throughput screening. Journal of Biomolecular Screening, 14(1), 66-76.

Conn, P. J., Jones, C. K., & Lindsley, C. W. (2009). Subtype-selective allosteric modulators of muscarinic receptors for the treatment of CNS disorders. Trends in Pharmacological Sciences, 30(3), 148-155.

Cornil, C. A. (2009). Rapid regulation of brain oestrogen synthesis: The behavioural roles of oestrogens and their fates. Journal of Neuroendocrinology, 21(3), 217-226.

Corona, G., Elia, C., Casetta, B., Diana, C., Rosalen, S., Bari, M., et al. (2009). A liquid chromatography-tandemmass spectrometry method for the simultaneous determination of exemestane and its metabolite 17-dihydroexemestane in human plasma. Journal of Mass Spectrometry, 44(6), 920-928.

Creton, R. (2009). Automated analysis of behavior in zebrafish larvae. Behavioural Brain Research, 203(1), 127-136.

D’Anglemont De Tassigny, X., Campagne, C., Steculorum, S., & Prevot, V. (2009). Estradiol induces physical association of neuronal nitric oxide synthase with NMDA receptor and promotes nitric oxide formation via estrogen receptor activation in primary neuronal cultures. Journal of Neurochemistry, 109(1), 214-224.

Damodaran, K., Nielsen, S. D., Geib, S. J., Zhang, W., Lu, Y., & Curran, D. P. (2009). Aryl-Csp3 bond rotation barriers of 2-aryl perhydropyrrolo[3,4- c]pyrrole-1,3-diones. Journal of Organic Chemistry, 74(15), 5481-5485.

Danot, O., Marquenet, E., Vidal-Ingigliardi, D., & Richet, E. (2009). Wheel of life, wheel of death: A mechanistic insight into signaling by STAND proteins. Structure, 17(2), 172-182.

de Azevedo Jr., W. F., Dias, R., Timmers, L. F. S. M., Pauli, I., Caceres, R. A., & Soares, M. B. P. (2009). Bioinformatics tools for screening of antiparasitic drugs. Current Drug Targets, 10(3), 232-239.

de Azevedo Jr., W. F., Caceres, R. A., Pauli, I., Timmers, L. F. S. M., Barcellos, G. B., Rocha, K. B., et al. (2009). Protein-drug interaction studies for development of drugs against plasmodium falciparum. Current Drug Targets, 10(3), 271-278.

de Kloe, G. E., Bailey, D., Leurs, R., & de Esch, I. J. P. (2009). Transforming fragments into candidates: Small becomes big in medicinal chemistry. Drug Discovery Today, 14(13-14), 630-646.

De Paoli, P. (2009). Institutional shared resources and translational cancer research. Journal of Translational Medicine, 7

De Wael, F., Jeanjot, P., Moens, C., Verbeuren, T., Cordi, A., Bouskela, E., et al. (2009). In vitro and in vivo studies of 6,8-(diaryl)imidazo[1,2-a]pyrazin-3(7H)-ones as new antioxidants. Bioorganic and Medicinal Chemistry, 17(13), 4336-4344.

Debotton, N., Giladi, O., Parnes, M., & Benita, S. (2009). Novel high-content paclitaxel palmitate nanospheres for improved cancer treatment. Journal of Drug Delivery Science and Technology, 19(4), 275-282.

Delomenède, M., Buchet, R., & Mebarek, S. (2009). Lansoprazole is an uncompetitive inhibitor of tissue-nonspecific alkaline phosphatase. Acta Biochimica Polonica, 56(2), 301-306.

Demian, D. J., Clugston, S. L., Foster, M. M., Rameh, L., Sarkes, D., Townson, S. A., et al. (2009). High-throughput, cell-free, liposome-based approach for assessing in vitro activity of lipid kinases. Journal of Biomolecular Screening, 14(7), 838-844.

Deshmukh, S. K., Mishra, P. D., Kulkarni-Almeida, A., Verekar, S., Sahoo, M. R., Periyasamy, G., et al. (2009). Anti-inflammatory and anticancer activity of ergoflavin isolated from an endophytic fungus. Chemistry and Biodiversity, 6(5), 784-789.

Diamond, M. S. (2009). Progress on the development of therapeutics against west nile virus. Antiviral Research, 83(3), 214-227.

Ding, X. -., Zhang, H. -., Qi, L., Zhao, B. -., Lian, S., Lv, H. -., et al. (2009). Synthesis of novel pyrazole carboxamide derivatives and discovery of modulators for apoptosis or autophagy in A549 lung cancer cells. Bioorganic and Medicinal Chemistry Letters, 19(18), 5325-5328.

Dissous, C., Ahier, A., & Long, T. (2009). A new promising drug against schistosomiasis. [Un nouvel espoir dans le traitement de la schistosomiase] Medecine/Sciences, 25(1), 24-26.

Doghman, M., & Lalli, E. (2009). A matter of dosage: SF-1 in adrenocortical development and cancer. Annales d’Endocrinologie, 70(3), 148-152.

dos Santos Filho, J. M., Leite, A. C. L., Oliveira, B. G. d., Moreira, D. R. M., Lima, M. S., Soares, M. B. P., et al. (2009). Design, synthesis and cruzain docking of 3-(4-substituted-aryl)-1,2,4-oxadiazole-N-acylhydrazones as anti-trypanosoma cruzi agents. Bioorganic and Medicinal Chemistry, 17(18), 6682-6691.

Drennan, M. B., Elewaut, D., & Hogquist, K. A. (2009). Thymic emigration: Sphingosine-1-phosphate receptor-1-dependent models and beyond. European Journal of Immunology, 39(4), 925-930.

Duerfeldt, A. S., Brandt, G. E. L., & Blagg, B. S. J. (2009). Design, synthesis, and biological evaluation of conformationally constrained cis-amide HSP90 inhibitors. Organic Letters, 11(11), 2353-2356.

Dunworth, W. P., & Caron, K. M. (2009). G protein-coupled receptors as potential drug targets for lymphangiogenesis and lymphatic vascular diseases. Arteriosclerosis, Thrombosis, and Vascular Biology, 29(5), 650-656.

Eglen, R. M., & Reisine, T. (2009). The current status of drug discovery against the human kinome. Assay and Drug Development Technologies, 7(1), 22-43.

Ekonomiuk, D., Su, X. -., Ozawa, K., Bodenreider, C., Siew, P. L., Otting, G., et al. (2009). Flaviviral protease inhibitors identified by fragment-based library docking into a structure generated by molecular dynamics. Journal of Medicinal Chemistry, 52(15), 4860-4868.

Ekonomiuk, D., Su, X. -., Ozawa, K., Bodenreider, C., Lim, S. P., Yin, Z., et al. (2009). Discovery of a non-peptidic inhibitor of west nile virus NS3 protease by high-throughput docking. PLoS Neglected Tropical Diseases, 3(1)

Ellmann, S., Sticht, H., Thiel, F., Beckmann, M. W., Strick, R., & Strissel, P. L. (2009). Estrogen and progesterone receptors: From molecular structures to clinical targets. Cellular and Molecular Life Sciences, 66(15), 2405-2426.

Emerson, C. H. (2009). Circulating thyroid stimulating hormones: Why, when, and what to measure. Thyroid, 19(1), 1-4.

Entzeroth, M., Flotow, H., & Condron, P. (2009). Overview of high-throughput screening. Current Protocols in Pharmacology, (SUPPL. 44), 9.4.1-9.4.27.

Ezgimen, M. D., Mueller, N. H., Teramoto, T., & Padmanabhan, R. (2009). Effects of detergents on the west nile virus protease activity. Bioorganic and Medicinal Chemistry, 17(9), 3278-3282.

Fehrenbacher, J. C., LoVerme, J., Clarke, W., Hargreaves, K. M., Piomelli, D., & Taylor, B. K. (2009). Rapid pain modulation with nuclear receptor ligands. Brain Research Reviews, 60(1), 114-124.

Fenton, R. A. (2009). Essential role of vasopressin-regulated urea transport processes in the mammalian kidney. Pflugers Archiv European Journal of Physiology, 458(1), 169-177.

Fisher, N., Warman, A. J., Ward, S. A., & Biagini, G. A. (2009). Chapter 17 type II NADH: Quinone oxidoreductases of plasmodium falciparum and mycobacterium tuberculosis. kinetic and high-throughput assays

Fix-Stenzel, S. R., Hayes, M. E., Zhang, X., Wallace, G. A., Grongsaard, P., Schaffter, L. M., et al. (2009). A stereoselective and scalable synthesis of a conformationally constrained S1P1 agonist. Tetrahedron Letters, 50(28), 4081-4083.

Foley, T. L., & Burkart, M. D. (2009). A homogeneous resonance energy transfer assay for phosphopantetheinyl transferase. Analytical Biochemistry, 394(1), 39-47.

Foss Jr., F. W., Mathews, T. P., Kharel, Y., Kennedy, P. C., Snyder, A. H., Davis, M. D., et al. (2009). Synthesis and biological evaluation of sphingosine kinase substrates as sphingosine-1-phosphate receptor prodrugs. Bioorganic and Medicinal Chemistry, 17(16), 6123-6136.

Fowler, R. A., Adhikari, N. K. J., Scales, D. C., Lee, W. L., & Rubenfeld, G. D. (2009). Update in critical care 2008. American Journal of Respiratory and Critical Care Medicine, 179(9), 743-758.

Fox, E. M., Andrade, J., & Shupnik, M. A. (2009). Novel actions of estrogen to promote proliferation: Integration of cytoplasmic and nuclear pathways. Steroids, 74(7), 622-627.

Franchi, L., Eigenbrod, T., Muñoz-Planillo, R., & Nuñez, G. (2009). The inflammasome: A caspase-1-activation platform that regulates immune responses and disease pathogenesis. Nature Immunology, 10(3), 241-247.

Franchi, L., Warner, N., Viani, K., & Nuñez, G. (2009). Function of nod-like receptors in microbial recognition and host defense. Immunological Reviews, 227(1), 106-128.

Fraser, I. D. C., & Germain, R. N. (2009). Navigating the network: Signaling cross-talk in hematopoietic cells. Nature Immunology, 10(4), 327-331.

Gao, J., Sidhu, S. S., & Wells, J. A. (2009). Two-state selection of conformation-specific antibodies. Proceedings of the National Academy of Sciences of the United States of America, 106(9), 3071-3076.

Gasparri, F. (2009). An overview of cell phenotypes in HCS: Limitations and advantages. Expert Opinion on Drug Discovery, 4(6), 643-657.

Gavrilyuk, J. I., Wuellner, U., Salahuddin, S., Goswami, R. K., Sinha, S. C., & Barbas III, C. F. (2009). An efficient chemical approach to bispecific antibodies and antibodies of high valency. Bioorganic and Medicinal Chemistry Letters, 19(14), 3716-3720.

George, S., Kumbhakar, M., Singh, P. K., Ganguly, R., Nath, S., & Pal, H. (2009). Fluorescence spectroscopic investigation to identify the micelle to gel transition of aqueous triblock copolymer solutions. Journal of Physical Chemistry B, 113(15), 5117-5127.

Gerber, A. N., Masuno, K., & Diamond, M. I. (2009). Discovery of selective glucocorticoid receptor modulators by multiplexed reporter screening. Proceedings of the National Academy of Sciences of the United States of America, 106(12), 4929-4934.

Gil, C., & Bräse, S. (2009). Solid-phase synthesis of biologically active benzoannelated nitrogen heterocycles: An update. Journal of Combinatorial Chemistry, 11(2), 175-197.

Gilbert, D. F., Wilson, J. C., Nink, V., Lynch, J. W., & Osborne, G. W. (2009). Multiplexed labeling of viable cells for high-throughput analysis of glycine receptor function using flow cytometry. Cytometry Part A, 75(5), 440-449.

Gossens, K., Naus, S., Corbel, S. Y., Lin, S., Rossi, F. M. V., Kast, J., et al. (2009). Thymic progenitor homing and lymphocyte homeostasis are linked via s1p-controlled expression of thymic p-selectin/ccl25. Journal of Experimental Medicine, 206(4), 761-778.

Graf, C., Rovina, P., & Bornancin, F. (2009). A secondary assay for ceramide kinase inhibitors based on cell growth inhibition by short-chain ceramides. Analytical Biochemistry, 384(1), 166-169.

Grigorova, I. L., Schwab, S. R., Phan, T. G., Pham, T. H. M., Okada, T., & Cyster, J. G. (2009). Cortical sinus probing, S1P1-dependent entry and flow-based capture of egressing T cells. Nature Immunology, 10(1), 58-65.

Guise, T. A., & Brown, S. A. (2009). Cancer treatment-related bone disease. Critical Reviews in Eukaryotic Gene Expression, 19(1), 47-60.

Habig, M., Blechschmidt, A., Dressler, S., Hess, B., Patel, V., Billich, A., et al. (2009). Efficient elimination of nonstoichiometric enzyme inhibitors from HTS hit lists. Journal of Biomolecular Screening, 14(6), 679-689.

Hakamata, W., Kurihara, M., Okuda, H., Nishio, T., & Oku, T. (2009). Design and screening strategies for α-glucosidase inhibitors based on enzymological information. Current Topics in Medicinal Chemistry, 9(1), 3-12.

Hammer, M. M., Kotecha, N., Irish, J. M., Nolan, G. P., & Krutzik, P. O. (2009). WebFlow: A software package for high-throughput analysis of flow cytometry data. Assay and Drug Development Technologies, 7(1), 44-55.

Hammond, R., Mauk, R., Ninaci, D., Nelson, D., & Gibbs, R. B. (2009). Chronic treatment with estrogen receptor agonists restores acquisition of a spatial learning task in young ovariectomized rats. Hormones and Behavior, 56(3), 309-314.

Han, G., Ma, H., Chintala, R., Fulton, D. J. R., Barman, S. A., & White, R. E. (2009). Essential role of the 90-kilodalton heat shock protein in mediating nongenomic estrogen signaling in coronary artery smooth muscle. Journal of Pharmacology and Experimental Therapeutics, 329(3), 850-855.

Hansch, C., & Verma, R. P. (2009). A QSAR study for the cytotoxic activities of taxoids against macrophage (MΦ)-like cells. European Journal of Medicinal Chemistry, 44(1), 274-279.

Hara, T., Hirasawa, A., Sun, Q., Sadakane, K., Itsubo, C., Iga, T., et al. (2009). Novel selective ligands for free fatty acid receptors GPR120 and GPR40. Naunyn-Schmiedeberg’s Archives of Pharmacology, 380(3), 247-255.

Harland, L., & Gaulton, A. (2009). Drug target central. Expert Opinion on Drug Discovery, 4(8), 857-872.

Hartung, H. -. (2009). New oral therapies may offer improved treatment options for patients with multiple sclerosis. Current Opinion in Neurology, 22(SUPPL. 1), S10-S14.

Hatae, J., Takami, N., Lin, H., Honda, A., & Inoue, R. (2009). 17β-estradiol-induced enhancement of estrogen receptor biosynthesis via MAPK pathway in mouse skeletal muscle myoblasts. Journal of Physiological Sciences, 59(3), 181-190.

Haynes, M. K., Strouse, J. J., Waller, A., Leitao, A., Curpan, R. F., Bologa, C., et al. (2009). Detection of intracellular granularity induction in prostate cancer cell lines by small molecules using the HyperCyt® high-throughput flow cytometry system. Journal of Biomolecular Screening, 14(6), 596-609.

He, M. -., Liu, L., Ge, W., Shaw, P. -., Jiang, R., Wu, L. -., et al. (2009). Antiangiogenic activity of tripterygium wilfordii and its terpenoids. Journal of Ethnopharmacology, 121(1), 61-68.

Hegedus, C., Szakács, G., Homolya, L., Orbán, T. I., Telbisz, Á, Jani, M., et al. (2009). Ins and outs of the ABCG2 multidrug transporter: An update on in vitro functional assays. Advanced Drug Delivery Reviews, 61(1), 47-56.

Herbst, K. J., Allen, M. D., & Zhang, J. (2009). The cAMP-dependent protein kinase inhibitor H-89 attenuates the bioluminescence signal produced by renilla luciferase. PLoS ONE, 4(5)

Herroeder, S., Reichardt, P., Sassmann, A., Zimmermann, B., Jaeneke, D., Hoeckner, J., et al. (2009). Guanine nucleotide-binding proteins of the G12 family shape immune functions by controlling CD4+ T cell adhesiveness and motility. Immunity, 30(5), 708-720.

Himanen, J. P., Goldgur, Y., Miao, H., Myshkin, E., Guo, H., Buck, M., et al. (2009). Ligand recognition by A-class eph receptors: Crystal structures of the EphA2 ligand-binding domain and the EphA2/ephrin-A1 complex. EMBO Reports, 10(7), 722-728.

Hiss, D. C., & Gabriels, G. A. (2009). Implications of endoplasmic reticulum stress, the unfolded protein response and apoptosis for molecular cancer therapy. part I: Targeting p53, Mdm2, GADD153/CHOP, GRP78/BiP and heat shock proteins. Expert Opinion on Drug Discovery, 4(8), 799-821.

Hollins, B., Kuravi, S., Digby, G. J., & Lambert, N. A. (2009). The c-terminus of GRK3 indicates rapid dissociation of G protein heterotrimers. Cellular Signalling, 21(6), 1015-1021.

Homma, K., Katagiri, K., Nishitoh, H., & Ichijo, H. (2009). Targeting ASK1 in ER stress-related neurodegenerative diseases. Expert Opinion on Therapeutic Targets, 13(6), 653-664.

Huang, X., Cao, J., & Huang, J. (2009). Solid-phase synthesis of benzofused tricycles based on benzimidazole from resin-bound 3-(2-aminophenylamino)-2-seleno-ester. Journal of Combinatorial Chemistry, 11(4), 515-518.

Hutter, M. C. (2009). In silico prediction of drug properties. Current Medicinal Chemistry, 16(2), 189-202.

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